{"product_id":"new-strategies-targeting-cancer-metabolism-anticancer-drugs-synthetic-analogues-and-antitumor-agents-paperback-9780128217832","title":"New Strategies Targeting Cancer Metabolism; Anticancer Drugs, Synthetic Analogues and Antitumor Agents (Paperback) 9780128217832","description":"\u003cfont face=\"Georgia\"\u003e\r\n\u003cp\u003e\u003cfont size=\"6\"\u003eNew Strategies Targeting Cancer Metabolism\u003c\/font\u003e\u003cbr\u003e\r\n\u003cfont size=\"5\"\u003eAnticancer Drugs, Synthetic Analogues and Antitumor Agents\u003c\/font\u003e\u003c\/p\u003e\r\n\r\n\u003cp\u003e\u003cem\u003ePresents up-to-date, synthetic strategies for the three main classes of antimetabolites integrated into various pharmaceutical agents\u003c\/em\u003e\u003c\/p\u003e\r\n\r\n\r\n\u003cp\u003e\u003cfont size=\"4\"\u003eGalal H. Elgemeie (Author), Reham A. Mohamed-Ezzat (Author)\u003c\/font\u003e\u003c\/p\u003e\r\n\r\n\u003cp\u003e\u003cfont size=\"3\"\u003e9780128217832, Elsevier Science\u003c\/font\u003e\u003c\/p\u003e\r\n\r\n\u003cp\u003e\u003cfont size=\"3\"\u003ePaperback, published 7 June 2022\u003c\/font\u003e\u003c\/p\u003e\r\n\r\n\u003cp\u003e\u003cfont size=\"3\"\u003e628 pages, Approx. 260 illustrations\u003cbr\u003e22.9 x 15.2 x 3.8 cm, 1.04 kg\u003c\/font\u003e\u003c\/p\u003e\r\n\r\n\r\n\r\n\r\n\r\n\u003cp align=\"justify\"\u003e\u003cstrong\u003e\u003cfont size=\"3\"\u003e\u003cp\u003e\u003ci\u003eNew Strategies Targeting Cancer Metabolism: Anticancer Drugs, Synthetic Analogues and Antitumor Agents\u003c\/i\u003e presents up-to-date synthetic strategies for three categories of antimetabolites: antifolates, purines and pyrimidines, the main classes of antimetabolites which are integrated into various pharmaceutical agents. Many of these antimetabolites are considered potent chemotherapeutic agents which have great potential impact on medical research. These main classes of antimetabolites are used in the treatment of critical diseases including cancer, malignancies, autoimmune diseases, and many other non-malignant diseases. Antineoplastic drugs such as alkylating agents which have significant effects are described. Novel synthetic strategies for many anticancer alkylating agents including nitrogen mustards, chlorambucil, melphalan, ifosamide, oxaliplatin and temozolomide are explored. Natural products have offered some of the most significant drugs for treating cancer, as many drugs currently in clinical use are derived from natural products as camptothecins, vinca alkaloids, and derivatives of podophyllotoxin. They provide a contribution that is essential for modern drug discovery and development. In this book, insights into a broad array of novel compounds are reviewed, well-recognized synthetic approaches are emphasized for further anticancer drug development and discovery, and the biological evaluation of novel synthesized compounds are included. This comprehensive reference is a valuable resource for medical chemists working in drug discovery and development, as well as pharmacologists and biochemists working in related fields.\u003c\/p\u003e\u003c\/font\u003e\u003c\/strong\u003e\u003c\/p\u003e\r\n\r\n\u003cp\u003e\u003cfont size=\"3\"\u003e\u003cp\u003e1. Medicinal chemistry of anticancer agents 2. Folate-based anticancer drugs 3. Purine-based anticancer drugs 4. Pyrimidine-based anticancer drugs 5. Synthetic strategies for anticancer antifolates 6. Synthetic strategies for purine nucleoside analogues 7. Synthetic strategies for pyrimidine nucleoside analogues 8. Anticancer alkylating agents 9. Natural products as anticancer agents 10. Synthetic strategies for antimetabolite analogues in our laboratory\u003c\/p\u003e\u003c\/font\u003e\u003c\/p\u003e\r\n\r\n\u003cp\u003e\u003cfont size=\"3\"\u003eSubject Areas: Organic chemistry [\u003ca title=\"See our other books on Organic chemistry\" href=\"https:\/\/freshlyprintedbooks.co.uk\/search?q=%22Organic%20chemistry%20%5BPNN%5D%22\"\u003ePNN\u003c\/a\u003e]\u003c\/font\u003e\u003c\/p\u003e\r\n\r\n\r\n\u003c\/font\u003e","brand":"Elsevier","offers":[{"title":"Default Title","offer_id":46650273923352,"sku":"9780128217832","price":151.29,"currency_code":"GBP","in_stock":false}],"thumbnail_url":"\/\/cdn.shopify.com\/s\/files\/1\/0730\/2037\/5320\/products\/9780128217832.jpg?v=1694107206","url":"https:\/\/freshlyprintedbooks.co.uk\/products\/new-strategies-targeting-cancer-metabolism-anticancer-drugs-synthetic-analogues-and-antitumor-agents-paperback-9780128217832","provider":"Freshly Printed Books","version":"1.0","type":"link"}